1u2o A 2.1 BS01 NEC A 1 A111 M154 N162 V197 Y200 A47 M90 N98 V127 Y130 ? 0005524,0006457,0016887,0051082,0140662 P41148 12970348 1001 GSHMLREKSEKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIGTSEFLNKMTEAQESTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTKTVWDWELMN 1u2o B 2.1 BS01 NEC B 1 A111 M154 N162 V197 Y200 A47 M90 N98 V127 Y130 ? 0005524,0006457,0016887,0051082,0140662 P41148 12970348 1002 GSHMLREKSEKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIGTSEFLNKMTEAQESTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTKTVWDWELMN 1ysz A 2.65 BS01 NEC A 1 A111 M154 N162 Y200 A38 M81 N89 Y121 ? 0005524,0006457,0016887,0051082,0140662 P41148 15951571 338 EKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIGTSEFLNKMTEAQESTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTKTVWDWELMN 2ydv A 2.6 BS01 NEC A 1 L85 T88 F168 N181 W246 L249 H250 N253 H278 L83 T86 F166 N179 W236 L239 H240 N243 H268 ? 0001609,0001973,0004930,0007186,0016020 Ki=16nM, IC50=3.7nM, EC50=251nM P29274 21593763 400 IMGSSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSAAAADILVGVLAIPFAIAISTGFCAACHGCLFIACFVLVLTASSIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCGQPKEGKAHSQGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQLKQMESQSTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFRKIIRSHVLRQQEPFKAAAAENLYFQ 5g53 A 3.4 BS01 NEC A 1 F168 E169 N181 W246 L249 H250 N253 M270 S277 H278 F151 E152 N164 W217 L220 H221 N224 M241 S248 H249 ? 0001609,0001973,0004930,0007186,0016020 Ki=16nM, IC50=3.7nM, EC50=251nM P29274 27462812 400 SSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADIAVGVLAIPFAITISTGFCAACHGCLFIACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQLKQMTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFRKIIRSHVLENLY 5g53 B 3.4 BS01 NEC B 1 F168 E169 N181 W246 L249 H250 N253 M270 S277 H278 F163 E164 N176 W225 L228 H229 N232 M249 S256 H257 ? 0001609,0001973,0004930,0007186,0016020 Ki=16nM, IC50=3.7nM, EC50=251nM P29274 27462812 400 SSVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADIAVGVLAIPFAITISTGFCAACHGCLFIACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCGQPKEGKAHSQGCGEGQVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTFRKIIRS 6b99 A 1.60238 BS01 NEC A 1 A55 M98 N106 F138 Y139 A40 M83 N91 F123 Y124 3.6.4.10 0005524,0006457,0016887,0051082,0140662 P07900 301 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVEKE 6d28 A 1.75 BS01 NEC A 1 A111 M154 N162 V197 Y200 A40 M83 N91 V126 Y129 ? 0005524,0006457,0016887,0051082,0140662 Kd=200nM P41148 12970348 401 KSEKFAFQAEVNRMMKLIINSLYKNKEIFLRELISNASDALDKIRLISLTDENALAGNEELTVKIKCDKEKNLLHVTDTGVGMTREELVKNLGTIAKSGTSEFLNKMTEAQEDGQSTSELIGQFGVGFYSAFLVADKVIVTSKHNNDTQHIWESDSNEFSVIADPRGNTLGRGTTITLVLKEEASDYLELDTIKNLVKKYSQFINFPIYVWSSKTKTVWDWELMN 6gdg A 4.11 BS01 NEC A 1 T88 Q89 M177 W246 L249 N253 M270 I274 H278 T82 Q83 M154 W211 L214 N218 M235 I239 H243 ? 0001609,0001973,0004930,0005515,0005737,0005829,0007186,0015035,0015036,0016020,0030337,0045454 P0AA25,P29274 29726815 400 AVYITVELAIAVLAILGNVLVCWAVWLNSNLQNVTNYFVVSLAAADIAVGVLAIPFAITISTGFCAACHGCLFIACFVLVLTQSSIFSLLAIAIDRYIAIRIPLRYNGLVTGTRAKGIIAICWVLSFAIGLTPMLGWNNCVACLFEDVVPMNYMVYFNFFACVLVPLLLMLGVYLRIFLAARRQLKQMTLQKEVHAAKSLAIIVGLFALCWLPLHIINCFTFFCPDCSHAPLWLMYLAIVLSHTNSVVNPFIYAYRIREFRQTF 7xy7 R 3.26 BS01 NEC R 1 T89 F173 M182 N186 M272 I276 S279 H280 T85 F152 M161 N165 M247 I251 S254 H255 ? 0001609,0001973,0002882,0004930,0005506,0005515,0005886,0007186,0007189,0007190,0009055,0010575,0010753,0016020,0019934,0020037,0022900,0032722,0032755,0042311,0042597,0043303,0043306,0045202,0046872,0060087,0098685,0098793,0098978,0099171 P0ABE7,P29275 36563137 501 TQDALYVALELVIAALSVAGNVLVCAAVGTANTLQTPTNYFLVSLAAADVAVGLFAIPFAITISLGFCTDFYGCLFLACFVLVLTQSSIFSLLAVAVDRYLAICVPLRYKSLVTGTRARGVIAVLWVLAFGIGLTPFLGWNSKDSALVKCLFENVVPMSYMVYFNFFGCVLPPLLIMLVIYIKIFLVACRQLQRTELRTTLQREIHAAKSLAMIVGIFALCWLPVHAVNCVTLFQPAQGKNKPKWAMNMAILLSHANSVVNPIVYAYRNRDFRYTFHKIISRY 8yh0 R 2.86 BS01 NEC R 1 T94 H95 F167 M176 I185 L245 N249 L263 H271 T86 H87 F159 M168 I177 L221 N225 L239 H247 0001609,0001973,0004930,0005886,0007186,0030425,0045202 A0A5P9VSM6,P03435,W5QED6 39511145 801 SWTSVTYITVEILIGLCAIVGNVLVIWVVKLNPSLQTTTFYFIVSLALADIAVGVLVMPLAIVISLGVTIHFYSCLFMTCLMLIFTHASIMSLLAIAVDRYLRVKLTVRYRRVTTQRRIWLALGLCWLVSFLVGLTPMFGWNMKLSSADENLTFLPCRFRSVMRMDYMVYFSFFLWILVPLVVMCAIYFDIFYIIRNRLEFKTAKSLLLVLFLFALCWLPLSIINCILYFDGQVPQTVLYLGILLSHANSMMNPIVYAYKIKKFKETYLLI