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GLASS

You can:

Go to the GPCR, ligand, or experimental data tables.
Go to the experimental data table for text mining information in PubMed ID column.
Go to the GPCR page and check other ligands which interact with it.
Go to the ligand page and check other GPCRs which it interacts with.
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GPCR

Name	Free fatty acid receptor 1
Species	Mus musculus (Mouse)
Gene	Ffar1
Synonym	FFA1 receptor FFA1R G protein-coupled receptor 40 G-protein coupled receptor 40 GPR40
Disease	N/A for non-human GPCRs
Length	300
Amino acid sequence	MDLPPQLSFALYVSAFALGFPLNLLAIRGAVSHAKLRLTPSLVYTLHLGCSDLLLAITLPLKAVEALASGAWPLPLPFCPVFALAHFAPLYAGGGFLAALSAGRYLGAAFPFGYQAIRRPRYSWGVCVAIWALVLCHLGLALGLETSGSWLDNSTSSLGINIPVNGSPVCLEAWDPDSARPARLSFSILLFFLPLVITAFCYVGCLRALVRSGLSHKRKLRAAWVAGGALLTLLLCLGPYNASNVASFINPDLGGSWRKLGLITGAWSVVLNPLVTGYLGTGPGRGTICVTRTQRGTIQK
UniProt	Q76JU9
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL5411
IUPHAR	N/A
DrugBank	N/A

Ligand

Name	CHEMBL229225
Molecular formula	C21H26O3
IUPAC name	3-[4-(2-ethylbutoxy)phenyl]-3-phenylpropanoic acid
Molecular weight	326.436
Hydrogen bond acceptor	3
Hydrogen bond donor	1
XlogP	5.1
Synonyms	SCHEMBL2949713 3-Aryl-3-(4-phenoxy)-propionic Acid derivative, 24 3-[4-(2-ethylbutoxy)phenyl]-3-phenylpropanoic acid BDBM22488
Inchi Key	VYGVLDBVEDZHAD-UHFFFAOYSA-N
Inchi ID	InChI=1S/C21H26O3/c1-3-16(4-2)15-24-19-12-10-18(11-13-19)20(14-21(22)23)17-8-6-5-7-9-17/h5-13,16,20H,3-4,14-15H2,1-2H3,(H,22,23)
PubChem CID	16738034
ChEMBL	CHEMBL229225
IUPHAR	N/A
BindingDB	22488
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand has a partition coefficient log P greater than 5.

Experimental Data

Parameter	Value	Reference	Database source
Activity	155.0 %	PMID17500511	ChEMBL
EC50	2200.0 nM	PMID17500511	ChEMBL

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