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BioLiP E. coli GLASS GPCR-HGmod GPCR-RD GPCR-EXP Tara-3D TM-fold DECOYS POTENTIAL RW/RWplus EvoEF HPSF THE-DB ADDRESS Alpaca-Antibody CASP7 CASP8 CASP9 CASP10 CASP11 CASP12 CASP13 CASP14

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GPCR

NameProteinase-activated receptor 2
SpeciesRattus norvegicus (Rat)
GeneF2rl1
Synonymcoagulation factor II (thrombin) receptor-like 1
coagulation factor II receptor-like 1
GPR11
PAR-2
PAR2
[ Show all ]
DiseaseN/A for non-human GPCRs
Length397
Amino acid sequenceMRSLSLAWLLGGITLLAASASCNRTVNAPGPNSKGRSLIGRLDTPPPITGKGAPVEPGFSVDEFSASVLTGKLTTVFLPVIYIIVFVIGLPSNGMALWVFFFRTKKKHPAVIYMANLALADLLSVIWFPLKISYHLHGNDWTYGDALCKVLIGFFYGNMYCSILFMTCLSVQRYWVIVNPMGHSRKRANIAVGVSLAIWLLIFLVTIPLYVMRQTIYIPALNITTCHDVLPEEVLVGDMFSYFLSLAIGVFLFPALLTASAYVLMIKTLRSSAMDEHSEKKRRRAIRLIITVLSMYFICFAPSNVLLVVHYFLIKSQRQSHVYALYLVALCLSTLNSCIDPFVYYFVSKDFRDQARNALLCRSVRTVKRMQISLTSNKFSRKSSSYSSSSTSVKTSY
UniProtQ63645
Protein Data BankN/A
GPCR-HGmod modelN/A
3D structure modelNo available structures or models
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLCHEMBL2429706
IUPHARN/A
DrugBankN/A

Known ligands

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Total entries: 5
Page:  / 1 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
391332D structureH-SER-PHE-LEU-LEU-ARG-NH2C30H51N9O6633.7958 / 9-0.5No
1729512D structureFSLLRY-NH2C39H60N10O8796.97110 / 110.6No
1893542D structureH-SER-PHE-LEU-LEU-ARG-OHC30H50N8O7634.7799 / 9-3.6No
2419102D structureCHEMBL2431726C29H56N10O7656.839 / 10-1.3No
3138282D structureSLIGRL-NH2C29H56N10O7656.839 / 10-1.3No

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