4hvs/2/1:A/2:A

Sequences
>4hvs-a2-m1-cA (length=326) [Search sequence]
HHMPMYEVQWKVVEESNGNNYSYIDPTQLPYDHKWEFPRNRLSFGKTLGAGAFGKVVEAT
AQGLIKSDAAMTVAVKMLKPSAHSTEREALMSELKVLSYLGNHENIVNLLGACTHGGPTL
VITEYCCYGDLLNFLRRKRDSFHSSDTSPASMEDDENALDLEDLLSFSYQVAKGMAFLAS
KNCIHRDLAARNILLTHGRITKICDFGLARDIKNDSNYVDKGNARLPVKWMAPESIFNSV
YTFESDVWSYGIFLWELFSLGSSPYPGMPVDSKFYKMIKEGFRMSSPEHAPAEMYDIMKT
CWDADPDKRPTFKQIVQDIEKQISES
>4hvs-a2-m2-cA (length=326) [Search sequence]
HHMPMYEVQWKVVEESNGNNYSYIDPTQLPYDHKWEFPRNRLSFGKTLGAGAFGKVVEAT
AQGLIKSDAAMTVAVKMLKPSAHSTEREALMSELKVLSYLGNHENIVNLLGACTHGGPTL
VITEYCCYGDLLNFLRRKRDSFHSSDTSPASMEDDENALDLEDLLSFSYQVAKGMAFLAS
KNCIHRDLAARNILLTHGRITKICDFGLARDIKNDSNYVDKGNARLPVKWMAPESIFNSV
YTFESDVWSYGIFLWELFSLGSSPYPGMPVDSKFYKMIKEGFRMSSPEHAPAEMYDIMKT
CWDADPDKRPTFKQIVQDIEKQISES
Structure information
PDB ID 4hvs (database links: RCSB PDB PDBe PDBj PDBsum)
Title Crystal structure of KIT kinase domain with a small molecule inhibitor, PLX647
Assembly ID 2
Resolution 1.9Å
Method of structure determination X-RAY DIFFRACTION
Number of inter-chain contacts 38
Sequence identity between the two chains 1.0
PubMed citation 23493555
Chain information
Chain 1 Chain 2
Model ID 1 2
Chain ID A A
UniProt accession P10721 P10721
Species 9606 (Homo sapiens) 9606 (Homo sapiens)
Function annotation BioLiP:4hvsA BioLiP:4hvsA
3D structure
Switch viewer: [NGL] [JSmol]
Dimer structure: Chain 1 in red; Chain 2 in blue.
Download: 4hvs-a2-m1-cA_4hvs-a2-m2-cA.pdb.gz
Full biological assembly
Download: 4hvs-assembly2.cif.gz

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