4qte/2/1:A/2:A |
| >4qte-a2-m1-cA (length=348) [Search sequence] |
PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLR EIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFL YQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVAT RWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQE DLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAH PYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY |
| >4qte-a2-m2-cA (length=348) [Search sequence] |
PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLR EIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFL YQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVAT RWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQE DLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAH PYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY |
|
| PDB ID |
4qte (database links:
RCSB PDB
PDBe
PDBj
PDBsum) |
| Title |
Structure of ERK2 in complex with VTX-11e, 4-{2-[(2-CHLORO-4-FLUOROPHENYL)AMINO]-5-METHYLPYRIMIDIN-4-YL}-N-[(1S)-1-(3-CHLOROPHENYL)-2-HYDROXYETHYL]-1H-PYRROLE-2-CARBOXAMIDE |
| Assembly ID |
2 |
| Resolution |
1.5Å |
| Method of structure determination |
X-RAY DIFFRACTION |
| Number of inter-chain contacts |
30 |
| Sequence identity between the two chains |
1.0 |
| PubMed citation |
25195011 |
|
|
Chain 1 |
Chain 2 |
| Model ID |
1 |
2 |
| Chain ID |
A |
A |
| UniProt accession |
P28482 |
P28482 |
| Species |
9606 (Homo sapiens) |
9606 (Homo sapiens) |
| Function annotation |
BioLiP:4qteA |
BioLiP:4qteA |
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Switch viewer: [NGL] [JSmol]
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Dimer structure:
Chain 1 in red;
Chain 2 in blue.
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Full biological assembly
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