4qte/2/1:A/2:A |
>4qte-a2-m1-cA (length=348) [Search sequence] |
PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLR EIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFL YQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVAT RWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQE DLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAH PYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY |
>4qte-a2-m2-cA (length=348) [Search sequence] |
PEMVRGQVFDVGPRYTNLSYIGEGAYGMVCSAYDNVNKVRVAIKKISPFEHQTYCQRTLR EIKILLRFRHENIIGINDIIRAPTIEQMKDVYIVQDLMETDLYKLLKTQHLSNDHICYFL YQILRGLKYIHSANVLHRDLKPSNLLLNTTCDLKICDFGLARVADPDHDHTGFLTEYVAT RWYRAPEIMLNSKGYTKSIDIWSVGCILAEMLSNRPIFPGKHYLDQLNHILGILGSPSQE DLNCIINLKARNYLLSLPHKNKVPWNRLFPNADSKALDLLDKMLTFNPHKRIEVEQALAH PYLEQYYDPSDEPIAEAPFKFDMELDDLPKEKLKELIFEETARFQPGY |
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PDB ID |
4qte (database links:
RCSB PDB
PDBe
PDBj
PDBsum) |
Title |
Structure of ERK2 in complex with VTX-11e, 4-{2-[(2-CHLORO-4-FLUOROPHENYL)AMINO]-5-METHYLPYRIMIDIN-4-YL}-N-[(1S)-1-(3-CHLOROPHENYL)-2-HYDROXYETHYL]-1H-PYRROLE-2-CARBOXAMIDE |
Assembly ID |
2 |
Resolution |
1.5Å |
Method of structure determination |
X-RAY DIFFRACTION |
Number of inter-chain contacts |
30 |
Sequence identity between the two chains |
1.0 |
PubMed citation |
25195011 |
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Chain 1 |
Chain 2 |
Model ID |
1 |
2 |
Chain ID |
A |
A |
UniProt accession |
P28482 |
P28482 |
Species |
9606 (Homo sapiens) |
9606 (Homo sapiens) |
Function annotation |
BioLiP:4qteA |
BioLiP:4qteA |
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Switch viewer: [NGL] [JSmol]
Dimer structure:
Chain 1 in red;
Chain 2 in blue.
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Full biological assembly
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