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Go to the GPCR, ligand, or experimental data tables.
Go to the experimental data table for text mining information in PubMed ID column.
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Go to the ligand page and check other GPCRs which it interacts with.
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GPCR

Name	Growth hormone secretagogue receptor type 1
Species	Rattus norvegicus (Rat)
Gene	Ghsr
Synonym	GH-releasing peptide receptor Ghrelin receptor ghrelin receptor 1a GHRP GHS-R growth hormone-releasing peptide receptor [ Show all ]
Disease	N/A for non-human GPCRs
Length	364
Amino acid sequence	MWNATPSEEPEPNVTLDLDWDASPGNDSLPDELLPLFPAPLLAGVTATCVALFVVGISGNLLTMLVVSRFRELRTTTNLYLSSMAFSDLLIFLCMPLDLVRLWQYRPWNFGDLLCKLFQFVSESCTYATVLTITALSVERYFAICFPLRAKVVVTKGRVKLVILVIWAVAFCSAGPIFVLVGVEHENGTDPRDTNECRATEFAVRSGLLTVMVWVSSVFFFLPVFCLTVLYSLIGRKLWRRRGDAAVGASLRDQNHKQTVKMLAVVVFAFILCWLPFHVGRYLFSKSFEPGSLEIAQISQYCNLVSFVLFYLSAAINPILYNIMSKKYRVAVFKLLGFESFSQRKLSTLKDESSRAWTKSSINT
UniProt	O08725
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL3278
IUPHAR	246
DrugBank	N/A

Ligand

Name	CHEMBL331303
Molecular formula	C36H47FN4O4
IUPAC name	(E)-5-amino-N-[(2R)-1-[[(2R)-3-(4-fluorophenyl)-1-[[(2R)-2-hydroxypropyl]amino]-1-oxopropan-2-yl]-methylamino]-1-oxo-3-(4-phenylcyclohexa-1,5-dien-1-yl)propan-2-yl]-N,5-dimethylhex-2-enamide
Molecular weight	618.794
Hydrogen bond acceptor	6
Hydrogen bond donor	3
XlogP	4.1
Synonyms	BDBM50066814 (E)-5-Amino-5-methyl-hex-2-enoic acid [(R)-1-{[(R)-2-(4-fluoro-phenyl)-1-((R)-2-hydroxy-propylcarbamoyl)-ethyl]-methyl-carbamoyl}-2-(4-phenyl-cyclohexa-1,5-dienyl)-ethyl]-methyl-amide
Inchi Key	ORUIITFKECREJK-YBTUSNJDSA-N
Inchi ID	InChI=1S/C36H47FN4O4/c1-25(42)24-39-34(44)31(22-27-15-19-30(37)20-16-27)41(5)35(45)32(40(4)33(43)12-9-21-36(2,3)38)23-26-13-17-29(18-14-26)28-10-7-6-8-11-28/h6-17,19-20,25,29,31-32,42H,18,21-24,38H2,1-5H3,(H,39,44)/b12-9+/t25-,29?,31-,32-/m1/s1
PubChem CID	44348031
ChEMBL	CHEMBL331303
IUPHAR	N/A
BindingDB	N/A
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand is heavier than 500 daltons.

Experimental Data

Parameter	Value	Reference	Database source
EC50	6.0 nM	PMID9733496	ChEMBL
Emax	90.0 %	PMID9733496	ChEMBL

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