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GPCR

NameNeuropeptide Y receptor type 1
SpeciesRattus norvegicus (Rat)
GeneNpy1r
SynonymFC5
neuropeptide Y receptor type 1
NPY-Y1 receptor
NPY1-R
Y1 receptor
[ Show all ]
DiseaseN/A for non-human GPCRs
Length382
Amino acid sequenceMNSTLFSRVENYSVHYNVSENSPFLAFENDDCHLPLAVIFTLALAYGAVIILGVSGNLALIIIILKQKEMRNVTNILIVNLSFSDLLVAVMCLPFTFVYTLMDHWVFGETMCKLNPFVQCVSITVSIFSLVLIAVERHQLIINPRGWRPNNRHAYIGITVIWVLAVASSLPFVIYQILTDEPFQNVSLAAFKDKYVCFDKFPSDSHRLSYTTLLLVLQYFGPLCFIFICYFKIYIRLKRRNNMMDKIRDSKYRSSETKRINVMLLSIVVAFAVCWLPLTIFNTVFDWNHQIIATCNHNLLFLLCHLTAMISTCVNPIFYGFLNKNFQRDLQFFFNFCDFRSRDDDYETIAMSTMHTDVSKTSLKQASPVAFKKISMNDNEKI
UniProtP21555
Protein Data BankN/A
GPCR-HGmod modelN/A
3D structure modelNo available structures or models
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLCHEMBL2587
IUPHAR305
DrugBankN/A

Known ligands

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Total entries: 17
Page:  / 1 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
513062D structureUNII-GLZ1WA47Q8C22H27Cl2N5O2464.3916 / 24.3Yes
710852D structureNPY2-36, porcineC181H278N54O554090.5462 / 58-17.7No
934912D structureNPY D-Trp32C196H290N56O56S4358.8765 / 59-15.6No
987572D structureBDBM85535C43H54N6O4S751.0037 / 36.2No
1558862D structureNPY, zebrafishC192H290N52O584254.7465 / 58-16.9No
1750122D structureBDBM50368404C112H174N36O272456.8533 / 41-3.6No
5541812D structureBIBP3226C27H31N5O3473.5774 / 52.5Yes
1856922D structureCHEMBL518564C31H45NaO5S552.7465 / 1N/ANo
1899262D structurePYY, zebrafishC194H292N52O574264.7864 / 56-15.5No
2978632D structure[125I]GW1229C110H170N34O242352.7848 / 386.8No
3142822D structureCHEMBL61532C30H41ClN4O2525.1345 / 15.7No
5549012D structureUNII-QKC82E736QC29H35N7O3529.6454 / 61.4No
3438542D structureNucleopeptide YC190H287N55O574253.7164 / 63-15.5No
3566782D structureL31,P34-NPY,humanC188H282N54O56S4226.7164 / 57-16.6No
5552572D structurehuman Neuropeptide YC189H285N55O57S4271.7565 / 63-16.2No
3950562D structureCHEMBL386823C57H91N17O121206.4615 / 16-0.6No
4393362D structureCHEMBL62166C27H24N4O3452.5144 / 23.4Yes

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